Chemical formula: C₂₅H₂₆F₆N₂O₂ Molecular mass: 500.485 g/mol PubChem compound: 10311306
Rolapitant is a selective antagonist of human substance P/neurokinin 1 (NK1) receptors.
This medicinal substance has been classified in the anatomical therapeutic chemical (ATC) classification according to its main therapeutic use as follows:
| ATC code | Group title | Classification |
|---|---|---|
| A04AD14 | A Alimentary tract and metabolism → A04 Antiemetics and antinauseants → A04A Antiemetics and antinauseants → A04AD Other antiemetics | |
Competent medicine agencies globally have authorized commercialization of this active ingredient according to these medication package inserts (MPIs):
| Title | Information Source | Document Type | |
|---|---|---|---|
| VARUBY Film-coated tablet | European Medicines Agency (EU) | MPI, EU: SmPC |
Rolapitant is an active ingredient of these brands:
United States (US)
Estonia (EE)
Lithuania (LT)
Poland (PL)
Note the following: The list of brand names is continuously updated, and thus does not include the total of products circulating worldwide. |
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