Teneligliptin

Chemical formula: C₂₂H₃₀N₆OS  Molecular mass: 426.22 g/mol  PubChem compound: 11949652

Active ingredient description

Teneligliptin is a potent, selective, and long-lasting DPP-4 inhibitor. It acts as a competitive reversible inhibitor of DPP-4 and decreases the degradation of incretins, especially GLP-1, thereby improving hyperglycemia by stimulating insulin secretion and suppressing glucagon secretion in a glucose-dependent manner (no or negligible risk of hypoglycemia).

Medicine classification

This medicinal substance has been classified in the anatomical therapeutic chemical (ATC) classification according to its main therapeutic use as follows:

ATC code Group title Classification
A10BH08 A Alimentary tract and metabolism → A10 Drugs used in diabetes → A10B Blood glucose lowering drugs, excl. insulins → A10BH Dipeptidyl peptidase 4 (DPP-4) inhibitors
Discover more medicines within A10BH08

Product monographs

Competent medicine agencies globally have authorized commercialization of this active ingredient according to these medication package inserts (MPIs):

Title Information Source Document Type  
TENEBLU Film-coated tablet Web Search MPI, Generic

Structural formula

Graphic representation of the active ingredient's molecular structure

External identifiers

CAS Substance: 760937-92-6
DrugBank Drug: DB11950
KEGG Drug: D08616
PubChem Compound: 11949652
SNOMED-CT Concept: 1172794002
Teneligliptin (substance)
UNII Identifier: 28ZHI4CF9C
TENELIGLIPTIN

Medicines

Teneligliptin is an active ingredient of these brands:

Japan (JP)

  • TENELIA as TENELIGLIPTIN HYDROBROMIDE HYDRATE

  • (combination) CANALIA as TENELIGLIPTIN HYDROBROMIDE HYDRATE

Nigeria (NG)

  • TENELISIGN as TENELIGLIPTIN HYDROBROMIDE HYDRATE

Note the following: The list of brand names is continuously updated, and thus does not include the total of products circulating worldwide.

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